MCHr1 antagonist 1

MCHr1antagonist1是一种选择性的黑色素浓集激素1型受体(melaninconcentratinghormone-1receptor)拮抗剂，对人MCH1受体的Kb和Ki值分别为1nM和4nM，在降低体重方面可能起作用。

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库存: 现货

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1mg

￥13550.00

10840.00

- +
5mg

￥27112.00

21690.00

- +
10mg

￥46087.00

36870.00

- +
20mg

￥81387.00

65110.00

- +

已选 0 种 0 瓶

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Background

MCHr1 antagonist 1 is a selective antagonist of melanin concentrating hormone-1 (MCH1) receptor, with a Kb of 1 nM and a Ki of 4 nM at human MCH1, and may be used to reduce the body mass.

MCHr1 antagonist 1 shows potent activities against melanin concentrating hormone-1 receptor, but less potent against human MCH1, NPY1, NPY5, GALR1, GALR2, GALR3, and rat 5HT2C receptors, with Kis of >50000 nM[1].

[1]. Selective melanin concentrating hormone-1 (MCH1) receptor antagonists and uses thereof. US 20030069261 A1