Methotrimeprazine (Levomepromazine) 是一种口服有效的抗精神病药物,通常用于在保守治疗中缓解恶心和呕吐。Methotrimeprazine (Levomepromazine) 对多种神经递质受体具有拮抗作用,包括多巴胺能、胆碱能、血清素和组胺受体。
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Methotrimeprazine (Levomepromazine) is an orally available neuroleptic agent, which is commonly used to relieve nausea and vomiting in palliative care settings. Levomepromazine has antagonist actions at multiple neurotransmitter receptor sites, including dopaminergic, cholinergic, serotonin and histamine receptors[1].
[1]. Cox L, et al. Levomepromazine for nausea and vomiting in palliative care. Cochrane Database Syst Rev. 2015 Nov 2;(11):CD009420. [2]. Sivaraman P, et al. Levomepromazine for schizophrenia. Cochrane Database Syst Rev. 2010 Oct 6;(10):CD007779.
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