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Ilorasertib hydrochloride
A multi-kinase inhibitor
(1E)-CFI-400437 dihydrochloride
CFI-400437 is a potent and selective polo-like kinase 4 (PLK4) inhibitor.
CD532 hydrochloride
An inhibitor of Aurora A kinase activity and the Aurora A-N-Myc protein-protein interaction
TL 13-12
TL 13-12 是一种有效的选择性 ALK-PROTAC 降解剂,可抑制 ALK 活性,IC50 值为 0.69 nM。 TL 13-12 还促进其他激酶的降解,包括 Aurora A、FER、PTK2 和 RPS6KA1,IC50 值分别为 13.5 nM、5.74 nM、18.4 nM 和 65 nM。 TL 13-12 由 TAE684 和 Pomalidomide 的 Cereblon 配体的缀合组成。
Histone H3 (21-44) (Phospho-Ser28) (human, mouse, rat, porcine, bovine) (trifluoroacetate salt)
A peptide fragment of histone H3
LY3295668 (AK-01)
LY3295668 (AK-01) is a potent, orally active and specific inhibitor of Aurora A kinase with Ki of 0.8 nM and 1038 nM for AURKA and AURKB, respectively.