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Bisindolylmaleimide XI (hydrochloride)
A PKC inhibitor
PKC β pseudosubstrate
Selective cell-permeable peptide inhibitor of protein kinase C
PKC-theta inhibitor
PKC-theta inhibitor (compound 20) inhibits PKC-θ with an IC50 of 18 nM.
PKC-IN-1
PKC-IN-1是一种有效的,ATP-竞争性的,可逆的PKC抑制剂,对人PKCβ和PKCα的Ki值分别为5.3和10.4nM,对人PKCα,PKCβI,PKCβII,PKCθ,PKCγ,PKCmu和PKCε的IC50值分别为2.3,8.1,7.6,25.6,57.5,314,808nM。
α-Amyloid Precursor Protein Modulator
α-Amyloid Precursor Protein Modulator 是一种细胞可渗透的苯并内酰胺衍生蛋白激酶 C (PKC) 激活剂,Ki 为 11.9 nM。
Dequalinium Chloride
An ammonium cation with diverse biological activities
Bisindolylmaleimide II
Bryostatin 2
Protein kinase C (PKC) activator
Bisindolylmaleimide III
PKC-9
A PKCζ inhibitor
VTX-27
A PKCθ inhibitor
1,2-Didecanoyl-sn-glycerol
An analog of DAG
PKCα (C2-4) Inhibitor Peptide
A PKCα inhibitor
3-Hydroxy Midostaurin-D5
3-Hydroxy Midostaurin-D5 (CGP52421-D5) 是 3-Hydroxy Midostaurin 的氘代化合物标准品。3-Hydroxy Midostaurin 是 PKC412 的代谢产物,可有效抑制 FMS 样酪氨酸激酶 3 (FLT3) 自磷酸化,在培养基和血浆中的 IC50 值分别约为 132 nM 和 9.8 μM。
(Des-octanoyl)-Ghrelin (human) (trifluoroacetate salt)
A peptide hormone