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Imrecoxib
Imrecoxib(BAP-909)艾瑞昔布是选择性环氧合酶 2 (COX-2) 抑制剂,IC50 值为 18 nM,也可以抑制 COX1 活性,IC50 值为 115 nM。Imrecoxib(BAP-909) 艾瑞昔布具有抗炎作用。
Thromboxane B1
The dihomo-γ-linolenic acid metabolite of COX/TXA synthase
Prostaglandin G2
The first stable intermediate in the COX pathway
Asaraldehyde
Asarylaldehyde (Asaronaldehyde) 是一种 COX-2 抑制剂,可显着抑制环氧合酶 II (COX-2) 的活性,IC50 值为 100 μg/mL。
Piroxicam
A COX inhibitor and NSAID
Diclofenac Sodium
An NSAID and a COX inhibitor
Prostaglandin D3
An inhibitor of platelet aggregation
Tenidap
A COX-1 selective NSAID
Lornoxicam
Fenbufen
An NSAID
Nabumetone
An NSAID and a prodrug form of 6-methoxy naphthalene acetic acid
Ketorolac
An NSAID and COX inhibitor
Rosmanol
A polyphenol with diverse biological activities
Ampiroxicam
A prodrug of piroxicam
Zaltoprofen
A non-selective COX inhibitor